Synthesis of thiazolidinones from 1,4-dithiocyanatobut …

Patel H. S, Mistry H. J, Desai H. D. Synthesis And Antimicrobial Activity Of Some New Thiazolidinones Containing N-Methyl Piperazine. Biosci Biotechnol Res Asia 2003;1(1). Available from:

Synthesis of Isoxazolyl Oxadiazolines and Thiazolidinones

SYNTHESIS, IN VITRO ANTIMICROBIAL ACTIVITY OF SCHIFF’S BASE, AZETIDINONES AND THIAZOLIDINONES

Synthesis of Bis-Thiazolidinones Using Chitosan …

Our previous study, based on a hybrid pharmacophore approach, allowed to establish a number of patterns in the structure–activity relationship (SAR) context for 4-thiazolidinones with a pyrazoline fragment in 2, 3 and 4 positions of the thiazolidone cycle, which possessed antitumor activity [7,8] .On the other hand, thiazolidinones and pyrazolines have occupied a unique position in the design and synthesis of novel biologically active agents that exert trypanocidal activity [9–13] .

Synthesis of piperazine-based thiazolidinones as …

Gupta, "Synthesis and Antimicrobial Profile of Newer Schiff Bases and Thiazolidinone Derivatives", WASET- International Journal of Chemical, Nuclear, Metallurgical and Materials Engineering, Vol.

Synthesis and evaluation of antimicrobial activity of thiazolidinone derivatives.

Doç. Dr. Ömer Faruk Bayrak | Yeditepe Üniversitesi …

N2 - 5-Arylidene-3-hydroxyalkyl-2-phenylimino-4-thiazolidinones (7,8) were synthesized and evaluated for their antidegenerative activity on human chondrocyte cultures stimulated by IL-1β. This in vitro model has proven to be a useful experimental model to reproduce the mechanisms involved in arthritic diseases. The cell viability, the amount of GAGs, the production of NO and PGE2 and the inhibition of MMP-3 were measured. Several thiazolidinones 7 and 8 exhibited the ability to block the production or action of the degenerative factors induced by IL-1β.

| Bioorganic & medicinal chemistry | …

T1 - Synthesis and in vitro evaluation of 5-arylidene-3-hydroxyalkyl-2-phenylimino-4-thiazolidinones with antidegenerative activity on human chondrocyte cultures

Synthesis and Antitubercular Activity of Some Novel Thiazolidinone Derivatives.

Synthesis and QSAR Studies on Thiazolidinones as Anti …

2. Vicini P., Geronikaki A. and et. Synthesis and antimicrobial activity of novel 2-tgiazolylimino-5-arylidene-4-thiazolidinones // Bioorganic and Medicinal Chemistry. – 2006. – Vol.14. –P.3859-3864.

Synthesis and antimicrobial evaluation of some novel 5-arylidine-3-aryl-Spiro[indane-thiazolidinone] derivatives

PDF Downloads : Oriental Journal of Chemistry

5-Arylidene-3-hydroxyalkyl-2-phenylimino-4-thiazolidinones (7,8) were synthesized and evaluated for their antidegenerative activity on human chondrocyte cultures stimulated by IL-1β. This in vitro model has proven to be a useful experimental model to reproduce the mechanisms involved in arthritic diseases. The cell viability, the amount of GAGs, the production of NO and PGE2 and the inhibition of MMP-3 were measured. Several thiazolidinones 7 and 8 exhibited the ability to block the production or action of the degenerative factors induced by IL-1β.

Design, synthesis and evaluation of thiazolidinone derivatives as antimicrobial and anti-viral agents.

2-mercaptopropionic acid, 79-42-5

AB - 5-Arylidene-3-hydroxyalkyl-2-phenylimino-4-thiazolidinones (7,8) were synthesized and evaluated for their antidegenerative activity on human chondrocyte cultures stimulated by IL-1β. This in vitro model has proven to be a useful experimental model to reproduce the mechanisms involved in arthritic diseases. The cell viability, the amount of GAGs, the production of NO and PGE2 and the inhibition of MMP-3 were measured. Several thiazolidinones 7 and 8 exhibited the ability to block the production or action of the degenerative factors induced by IL-1β.